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5VP0: DISCOVERY OF CLINICAL CANDIDATE N-{(1S)-1-[3-FLUORO-4- (TRIFLUOROMETHOXY)PHENYL]-2-METHOXYETHYL}-7-METHOXY-2-OXO-2,3- DIHYDROPYRIDO[2,3-B]PYRAZINE-4(1H)-CARBOXAMIDE (TAK-915), A HIGHLY POTENT, SELECTIVE, AND BRAIN-PENETRATING PHOSPHODIESTERASE 2A INHIBITOR FOR THE TREATMENT OF COGNITIVE DISORDERS
"cGMP-dependent 3',5'-cyclic phosphodiesterase" ( >99% identity ) with "BDBM50258896" ( exact match ):


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